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VYVANSE
Vyvanse, is the brand name for Lisdexamfetamine, a new
attention-deficit hyperactivity disorder (ADHD) drug. It received approval from
the U.S. Food and Drug Administration (FDA) on February 23, 2007.
Vyvanse Potential for Abuse?Vyvanse is intended to provide an option of lower abuse
potential. However, 50mg of Vyvanse contains 20mg of the stimulant d-amphetamine,
the well-known abusable Schedule II option. But because the key ingredient in
Vyvanse is bound to L-Lysine, the amphetamine is released at a slower rate in
the digestive system – as compared to Ritalin and Adderall. Therefore, Vyvanse
produced less "likeability", less euphoric effect and a later peak
time than amphetamine alone in clinical trials, suggesting that
lisdexamfetamine may be appropriate for use with patients with history of
stimulant abuse. Nevertheless, Vyvanse is currently up for designation as
Schedule II.
Schedule II drugs are known for their high abuse potential. Whether Vyvanse users will be able to find
other ways to abuse the drug, remains to be seen. Vyvanse Side EffectsThe most common side effects in studies of VYVANSE include: decreased appetite, difficulty falling asleep, stomachache, and
irritability.
According to the Vyvanse patent application, “These
compounds [found in Vyvanse] and compositions find particular use in providing
an abuse-resistant alternative treatment for certain disorders, such as
attention deficit hyperactivity disorder (ADHD), ADD, narcolepsy, and obesity.
Oral bioavailability of amphetamine is maintained at therapeutically useful
doses. At higher doses bioavailability is substantially reduced, thereby
providing a method of reducing oral abuse liability. Further, compounds and
compositions of the invention decrease the bioavailability of amphetamine by
parenteral routes, such as intravenous or intranasal administration, further
limiting their abuse liability.”
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